![]() ![]() Total Synthesis of Ripostatin B and Structure-Activity Relationship Studies on Ripostatin Analogs. Structural basis of small-molecule inhibition of human multidrug transporter ABCG2. A fluorescence anisotropy assay to discover and characterize ligands targeting the maytansine site of tubulin. The LAT1 inhibitor JPH203 reduces growth of thyroid carcinoma in a fully immunocompetent mouse model. Arylvinylpiperazine amides, a new class of potent inhibitors targeting QcrB of Mycobacterium tuberculosis. Studies toward the Total Synthesis of the Marine Macrolide Salarin C. Synthesis, Microtubule-Binding Affinity, and Antiproliferative Activity of New Epothilone Analogs and of an EGFR-Targeted Epothilone-Peptide Conjugate. Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands. Published online as an Accepted Article: external page call_made.ĩ8. Synthesis, Profiling and Bioactive Conformation of trans-Cyclopropyl Epothilones.
0 Comments
Leave a Reply. |
AuthorWrite something about yourself. No need to be fancy, just an overview. ArchivesCategories |